Using Thermal Shift Assays to Identify Inhibitors of the Isocitrate Lyase-1 Protein in Mycobacterium Tuberculosis

Session Number

Project ID: BIO 29

Advisor(s)

Dr. Angela Ahrendt; Illinois Mathematics and Science Academy

Discipline

Biology

Start Date

22-4-2020 10:25 AM

End Date

22-4-2020 10:40 AM

Abstract

Tuberculosis is an airborne respiratory disease that has a high latency period and is caused by the bacteria Mycobacterium tuberculosis. Nearly one third of the world’s population today is infected with this bacteria and approximately 1.3 million people experience tuberculosis related deaths every year. In this study, we chose to examine the isocitrate lyase-1 (ICL-1) protein as a possible target for the treatment of tuberculosis. We took this approach because ICL-1 allows the Mycobacterium tuberculosis bacteria to skip some of the steps in the KREBS cycle, which gives it the ability to survive in low-oxygen environments. The inhibition of ICL-1 could prevent the bacteria from becoming active within the human immune system. Different compounds were tested using a protein thermal shift assay to determine their efficacy in binding to the ICL-1 protein.

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Apr 22nd, 10:25 AM Apr 22nd, 10:40 AM

Using Thermal Shift Assays to Identify Inhibitors of the Isocitrate Lyase-1 Protein in Mycobacterium Tuberculosis

Tuberculosis is an airborne respiratory disease that has a high latency period and is caused by the bacteria Mycobacterium tuberculosis. Nearly one third of the world’s population today is infected with this bacteria and approximately 1.3 million people experience tuberculosis related deaths every year. In this study, we chose to examine the isocitrate lyase-1 (ICL-1) protein as a possible target for the treatment of tuberculosis. We took this approach because ICL-1 allows the Mycobacterium tuberculosis bacteria to skip some of the steps in the KREBS cycle, which gives it the ability to survive in low-oxygen environments. The inhibition of ICL-1 could prevent the bacteria from becoming active within the human immune system. Different compounds were tested using a protein thermal shift assay to determine their efficacy in binding to the ICL-1 protein.